What Makes an Oncology Therapy Practice-Changing?

Every year, hundreds of oncology studies are published and dozens of new therapies enter clinical development. Yet only a handful go on to change the standard of care. Why?

The answer isn’t simply that they are newer, more sophisticated, or based on a novel mechanism of action. Therapies that truly reshape oncology solve important clinical problems in ways that existing options don’t. They bring together compelling biology, thoughtful clinical development, meaningful patient benefit, and the ability to integrate into real-world care.

As oncology enters an era increasingly shaped by immunotherapies, antibody-drug conjugates (ADCs), radiopharmaceuticals, and precision medicines, the question is no longer simply, “Does this drug work?” It is also “Can it meaningfully change how patients are treated?” [1]

It Starts With an Unmet Medical Need

Practice-changing therapies begin by addressing problems that matter; demonstrating that value begins with clinical trial design.

Investigational therapies aim to extend survival where treatment options are limited, delay or prevent relapse, provide an effective option for patients with resistant disease, or reduce the burden of treatment without compromising outcomes. Therapies that deliver only incremental improvements—or enter disease settings already well served by existing treatments—face a higher bar for changing routine clinical practice.

Organizations such as ASCO have increasingly emphasized the importance of looking beyond statistical significance alone toward clinically meaningful benefit: improvements that translate into longer survival, better quality of life, more durable disease control, or other outcomes that matter to patients. [1-3]

This makes the choice of clinical trial endpoints critical. Endpoints establish the measurable benchmarks against which a therapy’s success or failure is evaluated and must therefore reflect both the outcomes that matter in a particular disease setting and the magnitude of benefit needed to be clinically meaningful within the evolving treatment landscape. These usually include overall survival (how long patients live), progression-free survival (how long patients live without their disease progressing), response rate (the proportion of patients whose tumors shrink by a predefined amount), duration of response (how long a treatment response is maintained), and patient-reported outcomes. Newer molecular measures, including minimal residual disease (MRD) in hematologic malignancies and circulating tumor DNA (ctDNA)-based detection of MRD in solid tumors, are also being explored—and, in certain settings, accepted—as earlier indicators of treatment benefit, reflecting a broader effort to identify endpoints that can generate meaningful evidence without waiting years for survival outcomes to mature.[4]

Meeting these benchmarks, however, establishes clinical trial success, not necessarily practice-changing potential. The magnitude of benefit must remain compelling in the context of the treatment landscape at the time the evidence emerges, while the overall risk-benefit profile must support a favorable regulatory decision.

Regulatory approval then enables a therapy to enter clinical practice, but does not by itself establish it as a standard of care. Depending on the healthcare system, subsequent reimbursement and health technology assessment decisions can determine the extent to which patients can access the therapy, while factors such as administration, monitoring, infrastructure, and treatment burden influence how readily it can be integrated into routine care. Together, these successive hurdles help determine whether an approved therapy is ultimately adopted into clinical practice.

Strong Biology Drives Better Development

The path toward becoming practice-changing begins long before a therapy reaches a pivotal clinical trial. A deep understanding of biology helps determine not only whether a therapeutic approach is scientifically defensible, but how it should be developed to generate the evidence needed to establish its place in clinical practice

A compelling biological rationale connects the therapeutic target or mechanism with the disease process, the intended patient population, and the expected clinical outcome. This understanding becomes particularly important as cancer evolves under treatment pressure and resistance mechanisms emerge.

Strong translational science can help answer critical questions early in development:

• Is the therapeutic mechanism relevant to the disease?
• Which patients are most likely to benefit?
• At what stage of disease should treatment be introduced?
• Which resistance mechanisms are likely to emerge?
• Could the therapy work more effectively in combination with another treatment?

The deeper the biological understanding, the more precisely these choices can be made.[3][4] Importantly, they are not simply R&D decisions: they shape the patient population, treatment setting, clinical endpoints, and ultimately the evidence against which a therapy will be judged relative to existing care.

The Right Therapy Needs the Right Patient

One of the critical lessons of modern oncology is that the effectiveness of a therapy can depend heavily on who receives it.

Precision oncology has demonstrated the value of matching treatments to molecular alterations, immune characteristics, or other features of tumor biology. Biomarker-driven patient selection can identify populations more likely to respond while helping spare others from treatments less likely to benefit them.

This has important implications not only for patient care, but for whether a therapy can demonstrate the magnitude of benefit needed to change practice. A therapy tested across a broad, biologically heterogeneous population may show only modest activity; in a well-defined population with the relevant disease biology, its effect may be substantially more pronounced.

Gefitinib, an oral targeted therapy, provides a landmark example: early studies in unselected patients with advanced non-small cell lung cancer (NSCLC) produced response rates of approximately 12-18%, while subsequent trials identified activating EGFR mutations as a stronger predictor of benefit. In the landmark IPASS study, the objective response rate among patients with EGFR-mutated tumors reached 71.2%, compared with just 1.1% among patients without an EGFR mutation. [5]

The difference illustrates how identifying the right patient population can transform the apparent clinical value of a therapy, and, in turn, its potential to change practice.[7]

Safety and Patient Experience Matter

Demonstrating meaningful efficacy in the right patient population is only part of the equation. For a therapy to change practice, the benefit it delivers must also justify the risks and practical demands associated with achieving it.

Evidently, safety is central to this assessment; the nature, severity, frequency, and reversibility of adverse events—as well as their impact on quality of life, treatment discontinuation, or the need for additional medical intervention—altogether influence the overall-risk benefit profile of a therapy. Importantly, what is considered acceptable depends on the clinical context: greater toxicity may be justified in an aggressive cancer with few effective options, while tolerance for the same risks may be considerably lower where effective and well-tolerated alternatives already exist.

For instance, despite their potentially life-threatening toxicities (including cytokine release syndrome and neurologic events), CAR-T therapies are reshaping the treatment of several hematologic malignancies, demonstrating how the acceptability of treatment related risk depends on the magnitude of clinical benefit, the disease setting, and the ability to manage those risk. Notably, in 2025, the FDA removed Risk Evaluation and Mitigation Strategy (REMS) requirements for six approved CAR-T therapies after concluding that the measures were no longer necessary to ensure their benefits outweighed their risks, illustrating how accumulating evidence and real-world clinical experience can change the benefit-risk assessment of a therapy and, in turn, its potential for broader clinical adoption.[6]

However, treatment burden extends beyond toxicity. Route and frequency of administration, time spent receiving treatment, monitoring requirements, hospital visits, and the need for specialist infrastructure all contribute to what receiving a therapy requires of patients and healthcare systems.[4][5] These considerations can extend beyond convenience: health technology assessments may explicitly account for administration costs, healthcare resource use, and the impact of treatment delivery on quality of life when evaluating a therapy’s overall value. Where these additional burdens materially affect cost-effectiveness relative to available alternatives, they can influence reimbursement decisions, the conditions under which a therapy is recommended, and ultimately how readily it is adopted into clinical practice.

Combinations Can Change What Existing Therapies Can Achieve

Practice-changing innovation does not always require replacing an established therapy. Increasingly, advances in oncology come from combining treatments in ways that extend what existing or emerging standards of care can achieve.

The biological rationale is compelling: cancer rarely depends on a single pathway, and tumors can adapt under therapeutic pressure. Rational combinations can target complementary mechanisms, overcome or delay resistance, deepen or prolong responses, or alter the tumor environment in ways that make an existing therapy more effective. In some cases, the interaction may be synergistic, meaning that the combined effect is greater than would be expected from the effects of the individual therapies alone.

A biologically compelling rationale, however, must translate into meaningful clinical benefit over the relevant treatment benchmark. Adding another agent can also add toxicity, treatment burden, complexity, and cost. To change practice, the combination must therefore demonstrate that the incremental benefit of adding the new therapy is sufficient to justify those additional demands.

This is why the most consequential combinations are not simply additive. Each component has a defined biological role, and the combination creates a clinically meaningful advantage over the established treatment backbone. When that happens, an investigational therapy does not need to displace the standard of care to change practice; it can change what the standard of care is capable of achieving.[8][9]

The Future Belongs to Thoughtful Innovation

As oncology expands into ADCs, radiopharmaceuticals, next-generation immunotherapies, cell therapies, and increasingly sophisticated combination approaches, scientific novelty alone will not determine which therapies ultimately reshape patient care.

Becoming practice-changing requires alignment across the development pathway: an important clinical problem, biology that supports the therapeutic approach, the right patient population and treatment setting, endpoints capable of demonstrating meaningful benefit, and a risk-benefit profile that remains compelling against an evolving standard of care. Beyond approval, access, treatment burden, and the practical realities of delivering therapy can further determine whether this potential translates into widespread clinical adoption.

Importantly, this assessment is not static and there is no universal threshold for what constitutes practice-changing benefit across oncology. Treatment landscapes evolve, new evidence emerges, and greater clinical experience can change how the benefits, risks, and practical value of a therapy are understood. A therapy may change practice by replacing an existing treatment, addressing a need for which no effective option exists, or making an established standard of care work better.

Ultimately, the most consequential innovation in oncology is not defined by novelty alone, but by the ability to translate scientific insight into a meaningful clinical benefit and, in doing so, change the standard of care.[11][12]

 

Bibliography

1. Gutierrez ME, Kummar S, Giaccone G. Next generation oncology drug development: opportunities and challenges. Nat Rev Clin Oncol. 2009;6(5):259-265. doi:10.1038/nrclinonc.2009.38

2. Rubin EH, Gilliland DG. Drug development and clinical trials–the path to an approved cancer drug. Nat Rev Clin Oncol. 2012;9(4):215-222. doi:10.1038/nrclinonc.2012.22

3. Dou YN, Grimstein C, Mascaro J, Wang J. Biomarkers for precision patient selection in cancer therapy approvals in the US, from 2011 to 2023. Clin Pharmacol Ther. 2024;116(2):304-314. doi:10.1002/cpt.3306

4. Fda.gov. Accessed August 11, 2026. https://www.fda.gov/vaccines-blood-biologics/safety-availability-biologics/fda-eliminates-risk-evaluation-and-mitigation-strategies-rems-autologous-chimeric-antigen-receptor

5. Sun JM, Won YW, Kim ST, et al. The different efficacy of gefitinib or erlotinib according to epidermal growth factor receptor exon 19 and exon 21 mutations in Korean non-small cell lung cancer patients. J Cancer Res Clin Oncol. 2011;137(4):687-694. doi:10.1007/s00432-010-0928-2

6. Fda.gov. Accessed August 11, 2026. https://www.fda.gov/regulatory-information/search-fda-guidance-documents/minimal-residual-disease-and-complete-response-multiple-myeloma-use-endpoints-support-accelerated

7. Moon DH, Chen RC. Defining a clinically meaningful benefit in cancer clinical trials: From the perspectives of the clinical trialist, patient, and society. JNCI Cancer Spectr. 2018;2(4):ky039. doi:10.1093/jncics/pky039

8. Real-world quantitative insights of cancer patient experience with subcutaneous (SC) vs intravenous (IV) drug delivery. ISPOR | International Society For Pharmacoeconomics and Outcomes Research. Accessed July 19, 2026. https://www.ispor.org/conferences-education/conferences/past-conferences/ispor-europe-2024/program/program/session/euro2024-4018/143383

9. de Miguel-Luken MJ, Mansinho A, Boni V, Calvo E. Immunotherapy-based combinations: current status and perspectives: Current status and perspectives. Curr Opin Oncol. 2017;29(5):382-394. doi:10.1097/CCO.0000000000000391

10. All-comers vs. Biomarker based patient selection for biotherapies in oncology- impact on drug development and market access. ISPOR | International Society For Pharmacoeconomics and Outcomes Research. Accessed July 19, 2026. https://www.ispor.org/heor-resources/presentations-database/presentation/ispor-europe-2018/all-comers-vs-biomarker-based-patient-selection-for-biotherapies-in-oncology-impact-on-drug-development-and-market-access

11. Mahmood I. Clinical pharmacology of antibody-drug conjugates. Antibodies (Basel). 2021;10(2):20. doi:10.3390/antib10020020

12. Riccardi F, Dal Bo M, Macor P, Toffoli G. A comprehensive overview on antibody-drug conjugates: from the conceptualization to cancer therapy. Front Pharmacol. 2023;14:1274088. doi:10.3389/fphar.2023.1274088

Jacek Antas

Chief Executive Officer


Jacek Antas is a shareholder of the Company, has spent more than 25 years in the financial services industry holding various positions in sales and consulting.

Mr. Antas obtained a master’s degree from the Warsaw School of Economics and has served as a board member of various
companies throughout his career.

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James B. Murphy

Chief Financial Officer


Mr. Murphy is a certified public accountant with over thirty years of experience in finance and operations management. He is currently a consultant with Danforth Advisors LLC (“Danforth”), a leading provider of outsourced strategic and operational specialists across functions in the life sciences industry. While at Danforth, Mr. Murphy has served over fifteen private and publicly held life sciences companies as CFO and CFO Advisor, helping them secure over USD 0.5 billion in financing and successfully execute pivotal asset transactions. Mr. Murphy functions as a consultant to Helix pursuant to a consulting agreement between the Company and Danforth.

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Thomas Mehrling

Medical Adviser


Thomas Mehrling (PhD in Pharmacology and MD) has over 20 years’ experience in multinational Pharma companies developing novel oncology compounds from preclinical research through to registration. Prior to entering the industry, he spent 13 years as an MD at the University Hospital in Frankfurt, working on preclinical and translational projects. He served as Director of European Oncology at Mundipharma International (2003–2013), building the company’s first European oncology business from the ground up out of Cambridge, UK, and completing the clinical development, registration and launch of two major products in Europe, DepoCyte® and Levact® (Ribomustin® and Treanda®). In 2013, he led the establishment of the Mundipharma Group’s start-up, Mundipharma EDO, developing anti-cancer therapeutics for solid tumours out of Basel, Switzerland.

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Kim Gaspar

Director Quality Assurance


Kim is the Director of Quality Assurance at Helix BioPharma Corp. An experienced quality assurance professional with expertise in Canadian, US, and EU regulations, she has been involved in all aspects of Phase I/II biopharmaceutical product development over the years, including regulatory submissions, QC laboratory compliance, tech transfer and third-party oversight of CMC activities, clinical QA, and bioanalytical data analysis. Kim joined Helix in 2000, transitioning into QA in 2003. She holds a B.Sc in Biochemistry and a Ph.D in Veterinary Physiological Sciences, both from the University of Saskatchewan.

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Brenda Lee

Director Clinical Operations


Brenda is the Clinical Operations Director at Helix Biopharma Corp. A clinical research operations professional with 25 years of experience managing clinical trials, ranging from early Phase I to late Phase IIIb/IV studies, she brings experience in clinical study protocol writing and development, trial start-up and vendor management, and a proven track record in planning and managing clinical trials to quality standards, timelines and budget. Brenda joined Helix Biopharma Corp. in 2018, working to advance the clinical program of L-DOS47. She holds B.Sc and M.Sc. degrees from the University of Toronto, specializing in Nutritional Sciences and Human Biology.

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Jerzy Leszczynski

Director


Jerzy Leszczynski is a shareholder of the Company, has spent more than 35 years developing businesses and has served in the capacity of board member of various real estate development companies. Mr. Leszczynski obtained his Master of Science in Chemistry from the Warsaw Institute of Technology.

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Janusz Grabski

Director, Chair of Audit Committee


Janusz (John) Grabski is a lawyer specialized in corporate and real estate law with over twenty years of experience.

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Malgorzata Laube

Director


Malgorzata Laube has over 19 years of experience in nuclear medicine. In her last role with Alberta Health Services, she was the Department Supervisor, Nuclear Medicine at Royal Alexandra Hospital. Ms. Laube obtained a MSc degree in Environmental Engineering from the Warsaw University of Technology and is based in Edmonton, Alberta, Canada.

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Jacek Antas

Chairman of the Board


Jacek Antas is a shareholder of the Company, has spent more than 25 years in the financial services industry holding various positions in sales and consulting.

Mr. Antas obtained a master’s degree from the Warsaw School of Economics and has served as a board member of various
companies throughout his career.

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Jonathan Davis

Advisor, ADC Discovery


Jonathan Davis received his Ph.D. from University of California, San Francisco, where he studied protein structure and function using NMR. After a post-doc at Harvard Medical School exploring RNA selection and structure in the labs of Jack Szostak and Gerhard Wagner, he went to work at EMD Serono, where his work involved improving antibody-based therapeutics, inventing a platform technology for generating heterodimeric Fcs as a basis for multifunctional molecules, and developing a novel scaffold based on an artificially-designed protein from David Baker’s lab. In 2008 he took a job at Bristol-Myers Squibb in Waltham/Cambridge MA, working on antibody discovery and platform development in a wide range of therapeutic areas, with a particular focus on multispecific therapeutics. He moved to Madison, WI in 2019 to take on the role of VP of Innovation and Strategy at Invenra, a biotech focused on bispecific antibodies, and where he is currently head of the Scientific Advisory Board. In early 2024 he left the corporate world to found Creative Antibodies, a consulting firm that helps guide companies to successful antibody discovery and development projects, from mAbs to multispecifics, ADCs, and other formats. Outside of science, Jonathan is a conservatory trained cellist, plays numerous other instruments, and founded the UCSF Orchestra (now Symphony Parnassus) in San Francisco, where he was Music Director for six years.

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Davide Guggi

Advisor, CMC


Davide graduated as a pharmacist and received his PhD in Pharmaceutical Technology and Biotechnology from the University of Vienna. He has over 20 years of experience in the pharmaceutical industry, principally in the field of oncology. At the beginning of his career, Davide led oncology business units and commercial departments at Mundipharma and Gilead across Austria and Eastern Europe. Since over 10 years he has been working as a CMC expert, covering operational and regulatory CMC functions on behalf of over 20 different small- and medium-sized biotech companies across the world. He has served as CMC Director and CSO/CTO for several years, developing both small molecules and biologics (mABs, Fab, ADCs and Radio-immuno-conjugates) from early discovery to NDA/BLA in the US, EU and Canada, with a focus on First-in-Human and Phase I/II studies in oncology indications.

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Tumor Defense Breaker™, L-DOS47


L‑DOS47 is a first‑in‑class, clinical-stage antibody‑enzyme conjugate designed to deliver a game-changing assist to anti-cancer immunity and today’s leading cancer immunotherapies for the treatment of prevalent, hard-to-treat solid tumors. The compound precisely targets CEACAM6, a cell-surface protein overexpressed in non‑small cell lung cancer (NSCLC) and other aggressive tumors, where it delivers an enzymatic payload that raises the extracellular pH of the acidic tumor microenvironment (TME). By neutralizing tumor acidity, L-DOS47 restores immune cell infiltration and activity, helps turn immunologically “cold” tumors “hot”, and enhances the therapeutic reach of immune checkpoint inhibitors. With patented composition-of-matter coverage through 2036 and demonstrated synergy with PD-1 inhibitor, pembrolizumab, L-DOS47 is poised to significantly increase the efficacy of immune checkpoint blockade and unlock broader and more durable responses in NSCLC and other aggressive solid tumors.

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LEUMUNA™


LEUMUNA™ is an oral immune checkpoint modulator designed to activate the donor immune system to recognize and fight relapsing leukemia in patients who have undergone allogeneic stem cell transplantation (allo-SCT). Although a life-saving procedure, up to 30% of patients who undergo allo-SCT see their cancer return, facing a median survival of just four months. LEUMUNA aims to offer these patients a new lease on life, by activating an immune cascade and inciting graft-versus-leukemia (GvL) effect, potentially offering long-term remission. Backed by strong preclinical data and a promising safety record from trials with its precursor compound, ulodesine, LEUMUNA offers a patient‑friendly, oral approach to a difficult-to-treat condition, with patent protection through 2041 and an Orphan Drug Designation granted by the US FDA.

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GEMCEDA™


GEMCEDA is a first-in-class oral prodrug of gemcitabine that opens up the possibility for convenient at-home administration, metronomic dosing and seamless integration into combination regimens with immune checkpoint inhibitors. To date, gemcitabine is only administered intravenously because oral forms have shown poor bioavailability of about 10%. GEMCEDA was developed as a prodrug to enable new uses of gemcitabine by combining it with cedazuridine, an enzyme inhibitor that helps boost its bioavailability to 90%. This remarkable innovation allows for greater flexibility in dosing schedules, fewer clinic visits, and a better quality of life, while achieving bioavailability on par with intravenous gemcitabine. Supported by a well‑established safety profile, scalable manufacturing, and patent coverage to 2043, GEMCEDA reimagines how chemotherapy can fit into patients’ lives.

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